Prashant R. Murumkar: search on Z-Library

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1

Identifying the structural features and diversifying the chemical domain of peripherally acting CB1 receptor antagonists using molecular modeling techniques

Sharma, Mayank Kumar, Murumkar, Prashant, Kuang, Guanglin, Tang, Yun, Yadav, Mange Ram

Journal:

Year:

2015

Language:

english

File:

PDF, 2.08 MB

english, 2015

2

One-pot synthesis, biological evaluation, and docking study of new chromeno-annulated thiopyrano[2,3-c]pyrazoles

Parmar, Bhagyashri D., Sutariya, Tushar R., Brahmbhatt, Gaurangkumar C., Parmar, Narsidas J., Kant, Rajni, Gupta, Vivek K., Murumkar, Prashant R., Sharma, Mayank Kumar, Yadav, Mange Ram

Journal:

Molecular Diversity

Year:

2016

Language:

english

File:

PDF, 1.90 MB

english, 2016

3

New role of phenothiazine derivatives as peripherally acting CB1 receptor antagonizing anti-obesity agents

Sharma, Mayank Kumar, Machhi, Jatin, Murumkar, Prashant, Yadav, Mange Ram

Journal:

Scientific Reports

Year:

2018

Language:

english

File:

PDF, 2.30 MB

english, 2018

4

Vicinal Diaryl Substituted Heterocycles || Vicinal Diaryl Oxadiazoles, Oxazoles, and Isoxazoles

Murumkar, Prashant R.

Year:

2018

Language:

english

File:

PDF, 840 KB

english, 2018

5

LIGANDS OF THE CORE ACETYLCHOLINE BIOSYNTHESIZING ENZYME, CHOLINE ACETYLTRANSFERASE, AS NOVEL AND POTENTIAL THERAPEUTIC AGENTS AND IN VIVO PET TRACERS FOR EARLY DIAGNOSIS OF ALZHEIMERâS DISEASE

Darreh-Shori, Taher, Kumar, Rajnish, Kumar, Amit, Murumkar, Prashant, Nag, Sangram, Jia, Zhisheng, Arakawa, Ryosuke, Leuzy, Antoine, Lemoine, Laetitia, Nordberg, Agneta, Yadav, Mange Ram, Halldin, Chr

Journal:

Alzheimer's & Dementia

Year:

2019

File:

PDF, 120 KB

2019

6

Current perspective of TACE inhibitors: A review

Shirshendu DasGupta, Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 809 KB

english, 2009

7

Studies on novel 2-imidazolidinones and tetrahydropyrimidin-2(1H)-ones as potential TACE inhibitors: Design, synthesis, molecular modeling, and preliminary biological evaluation

Shirshendu DasGupta, Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 1.34 MB

english, 2009

8

Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists—A perspective

Prashant Naik, Prashant Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 6.83 MB

english, 2010

9

Development of highly predictive 3D-QSAR CoMSIA models for anthraquinone and acridone derivatives as telomerase inhibitors targeting G-quadruplex DNA telomere

Vishal P. Zambre, Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Journal of Molecular Graphics and Modelling

Year:

2010

Language:

english

File:

PDF, 513 KB

english, 2010

10

Development of predictive pharmacophore model for in silico screening, and 3D QSAR CoMFA and CoMSIA studies for lead optimization, for designing of potent tumor necrosis factor alpha converting enzyme inhibitors

Prashant Revan Murumkar, Vishal Prakash Zambre, Mange Ram Yadav

Journal:

Journal of Computer-Aided Molecular Design

Year:

2010

Language:

english

File:

PDF, 1.49 MB

english, 2010

11

3D-Quantitative Structure–Activity Relationship Studies on Benzothiadiazepine Hydroxamates as Inhibitors of Tumor Necrosis Factor-α Converting Enzyme

Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav

Journal:

Chemical Biology & Drug Design

Year:

2008

Language:

english

File:

PDF, 482 KB

english, 2008

12

Development of Predictive 3D-QSAR CoMFA and CoMSIA Models for β-aminohydroxamic Acid-Derived Tumor Necrosis Factor-α Converting Enzyme Inhibitors

Prashant R. Murumkar, Shirshendu Das Gupta, Vishal P. Zambre, Rajani Giridhar, Mange Ram Yadav

Journal:

Chemical Biology & Drug Design

Year:

2009

Language:

english

File:

PDF, 498 KB

english, 2009

13

Synthesis, preliminary biological evaluation and molecular modeling of some new heterocyclic inhibitors of TACE

Prabal Sengupta, Chetan S. Puri, Hemant A. Chokshi, Chetana K. Sheth, Ajay S. Midha, Trinadha Rao Chitturi, Rajamannar Thennati, Prashant R. Murumkar, Mange Ram Yadav

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 428 KB

english, 2011

14

Novel methods and strategies in the discovery of TACE inhibitors

Murumkar, Prashant R, Giridhar, Rajani, Yadav, Mange Ram

Journal:

Expert Opinion on Drug Discovery

Year:

2013

Language:

english

File:

PDF, 1020 KB

english, 2013

15

Three-dimensional quantitative structure–activity relationship CoMFA/CoMSIA on pyrrolidine-based tartrate diamides as TACE inhibitors

Prashant R. Murumkar, Mayank Kumar Sharma, Anurag C. Shinde…

Journal:

Medicinal Chemistry Research

Year:

2013

Language:

english

File:

PDF, 527 KB

english, 2013

16

Synthesis and investigation of anti-inflammatory activity of novel nitric oxide donating hybrid drugs

Shailesh L. Chandak, Amol S. Bansode, Prashant R. Murumkar…

Journal:

Medicinal Chemistry Research

Year:

2013

Language:

english

File:

PDF, 602 KB

english, 2013

17

Novel TACE inhibitors in drug discovery: a review of patented compounds

Murumkar, Prashant R, DasGupta, Shirshendu, Chandani, Sneha R, Giridhar, Rajani, Yadav, Mange Ram

Journal:

Expert Opinion on Therapeutic Patents

Year:

2010

Language:

english

File:

PDF, 785 KB

english, 2010

18

Determination of structural requirements of influenza neuraminidase type A inhibitors and binding interaction analysis with the active site of A/H1N1 by 3D-QSAR CoMFA and CoMSIA modeling

Murumkar, Prashant R., Le, Ly, Truong, Thanh N., Yadav, Mange Ram

Journal:

Year:

2011

Language:

english

File:

PDF, 429 KB

english, 2011

19

Prospective therapeutic agents for obesity: Molecular modification approaches of centrally and peripherally acting selective cannabinoid 1 receptor antagonists

Sharma, Mayank Kumar, Murumkar, Prashant R., Kanhed, Ashish M., Giridhar, Rajani, Yadav, Mange Ram

Journal:

European Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 11.28 MB

english, 2014

20

Synthesis and biological evaluation of some novel pyrido[1,2-a]pyrimidin-4-ones as antimalarial agents

Mane, Uttam R., Mohanakrishnan, D., Sahal, Dinkar, Murumkar, Prashant R., Giridhar, Rajani, Yadav, Mange Ram

Journal:

European Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 2.47 MB

english, 2014

21

Structural Investigations of Acridine Derivatives by CoMFA and CoMSIA Reveal Novel Insight into Their Structures toward DNA G-Quadruplex Mediated Telomerase Inhibition and Offer a Highly Predictive 3D-Model for Substituted Acridines

Zambre, Vishal P., Murumkar, Prashant R., Giridhar, Rajani, Yadav, Mange Ram

Journal:

Journal of Chemical Information and Modeling

Year:

2009

Language:

english

File:

PDF, 6.21 MB

english, 2009

22

Virtual screening-based identification of lead molecules as selective TACE inhibitors

Murumkar, Prashant R., Sharma, Mayank Kumar, Giridhar, Rajani, Yadav, Mange Ram

Journal:

Medicinal Chemistry Research

Year:

2015

Language:

english

File:

PDF, 1.63 MB

english, 2015

23

A comprehensive patents review on cannabinoid 1 receptor antagonists as antiobesity agents

Sharma, Mayank Kumar, Murumkar, Prashant R, Barmade, Mahesh A, Giridhar, Rajani, Yadav, Mange Ram

Journal:

Expert Opinion on Therapeutic Patents

Year:

2015

Language:

english

File:

PDF, 3.77 MB

english, 2015

24

Exploring structural requirements for peripherally acting 1,5-diaryl pyrazole-containing cannabinoid 1 receptor antagonists for the treatment of obesity

Sharma, Mayank Kumar, Murumkar, Prashant R., Giridhar, Rajani, Yadav, Mange Ram

Journal:

Molecular Diversity

Year:

2015

Language:

english

File:

PDF, 3.82 MB

english, 2015

25

3-Substituted 1-methyl-3-benzazepin-2-ones as 5-HT 2C receptor agonists

Shidore, Mahesh, Machhi, Jatin, Murumkar, Prashant, Barmade, Mahesh, Thanki, Jigar, Yadav, Mange Ram

Journal:

Year:

2015

Language:

english

File:

PDF, 844 KB

english, 2015

26

Exploration of 6,7-dimethoxyquinazoline derivatives as dual acting α1- and AT1-receptors antagonists: Synthesis, evaluation, pharmacophore & 3D-QSAR modeling and receptor docking studies

Agrawal, Neetesh Kumar, Machhi, Jatin, Rathwa, Virendra, Kanhed, Ashish, Patel, Sagar, Murumkar, Prashant, Gandhi, Hardik, Yadav, Mange Ram

Journal:

Year:

2016

Language:

english

File:

PDF, 2.29 MB

english, 2016

27

A catalyst− and solvent−free multicomponent synthesis and docking study of some new antiproliferative N5-allyl-quinolylpyrido [2,3-b][1,4] benzodiazepinone precursors

PARMAR, NARSIDAS JERAMDAS, Barad, Hitesh A, Sutariya, Tushar R, Brahmbhatt, Gaurangkumar C., Lagunes, Irene, Padron, Jose M, Murumkar, Prashant, Sharma, Mayank, Yadav, Mange Ram

Journal:

New Journal of Chemistry

Year:

2016

Language:

english

File:

PDF, 1009 KB

english, 2016

28

Benzylpiperidine-linked diarylthiazoles as potential anti-Alzheimer’s agents-synthesis and biological evaluation

Shidore, Mahesh, Machhi, Jatin, Shingala, Kaushik, Murumkar, Prashant, Sharma, Mayank Kumar, Agrawal, Neetesh, Tripathi, Ashutosh, Parikh, Zalak, Pillai, Prakash, Yadav, Mange Ram

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 3.24 MB

english, 2016

29

Contemporary developments in the discovery of selective factor Xa inhibitors: A review

Patel, Nirav R., Patel, Dushyant V., Murumkar, Prashant R., Yadav, Mange Ram

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.73 MB

english, 2016

30

ChemInform Abstract: Developing Steroidal Aromatase Inhibitors - An Effective Armament to Win the Battle Against Breast Cancer

Yadav, Mange Ram, Barmade, Mahesh A., Tamboli, Riyaj S., Murumkar, Prashant R.

Journal:

Year:

2015

File:

PDF, 12 KB

2015

31

ChemInform Abstract: Prospective Therapeutic Agents for Obesity: Molecular Modification Approaches of Centrally and Peripherally Acting Selective Cannabinoid 1 Receptor Antagonists

Sharma, Mayank Kumar, Murumkar, Prashant R., Kanhed, Ashish M., Giridhar, Rajani, Yadav, Mange Ram

Journal:

Year:

2014

File:

PDF, 17 KB

2014

32

Dihydropyrimidinone-isatin hybrids as novel non-nucleoside HIV-1 reverse transcriptase inhibitors

Devale, Titiksh L., Parikh, Jignesh, Miniyar, Pankaj, Sharma, Pankaj, Shrivastava, Birendra, Murumkar, Prashant

Journal:

Bioorganic Chemistry

Year:

2017

Language:

english

File:

PDF, 2.03 MB

english, 2017

33

Vicinal diaryl azole-based urea derivatives as potential cholesterol lowering agents acting through inhibition of SOAT enzymes

Pal, Palash, Gandhi, Hardik P., Kanhed, Ashish M., Patel, Nirali R., Mankadia, Niraj N., Baldha, Satish N., Barmade, Mahesh A., Murumkar, Prashant R., Yadav, Mange Ram

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 2.00 MB

english, 2017

34

ChemInform Abstract: Contemporary Developments in the Discovery of Selective Factor Xa Inhibitors: A Review

Patel, Nirav R., Patel, Dushyant V., Murumkar, Prashant R., Yadav, Mange Ram

Journal:

Year:

2016

File:

PDF, 14 KB

2016

35

An Overview of the Development of DprE1 Inhibitors for Combating the Menace of Tuberculosis

Chikhale, Rupesh Vitthalrao, Barmade, Mahesh A., Murumkar, Prashant R., Yadav, Mange Ram

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.56 MB

english, 2018

36

Vicinal Diaryl Substituted Heterocycles || Vicinal Diaryl Triazoles and Tetrazoles

Murumkar, Prashant R.

Year:

2018

Language:

english

File:

PDF, 2.10 MB

english, 2018

37

Advances in patented CB1 receptor antagonists for obesity

Yadav, Mange Ram, Murumkar, Prashant R

Journal:

Pharmaceutical Patent Analyst

Year:

2018

Language:

english

File:

PDF, 322 KB

english, 2018

38

Drug-fortified liposomes as carriers for sustained release of NSAIDs: The concept and its validation in the animal model for the treatment of arthritis

Pawar, Vijay A., Manjappa, Arehalli S., Murumkar, Prashant R., Gajaria, Tejal K., Devkar, Ranjisinh V., Mishra, Anil K., Yadav, Mange Ram

Journal:

European Journal of Pharmaceutical Sciences

Year:

2018

Language:

english

File:

PDF, 7.23 MB

english, 2018

39

Gemini Amphiphile-Based Lipoplexes for Efficient Gene Delivery: Synthesis, Formulation Development, Characterization, Gene Transfection, and Biodistribution Studies

Yadav, Mange R., Kumar, Mukesh, Murumkar, Prashant R., Hazari, Puja P., Mishra, Anil K.

Journal:

Year:

2018

Language:

english

File:

PDF, 4.81 MB

english, 2018

40

DISCOVERY OF NOVEL SMALL MOLECULES FOR THE TREATMENT OF ALZHEIMER'S DISEASE

Murumkar, Prashant R., Yadav, Mange Ram, Darreh-Shori, Taher, Kumar, Amit, Kumar, Rajnish

Journal:

Alzheimer's & Dementia

Year:

2019

Language:

english

File:

PDF, 119 KB

english, 2019

41

Recent developments and strategies for the discovery of TACE inhibitors

Murumkar, Prashant R., Ghuge, Rahul B., Chauhan, Monica, Barot, Rahul R., Sorathiya, Sharmishtha, Choudhary, Kailash M., Joshi, Karan D., Yadav, Mange Ram

Journal:

Expert Opinion on Drug Discovery

Year:

2020

File:

PDF, 3.31 MB

2020

42

P3-108: CHAT POTENTIATING LIGANDS (CPLS): A NOVEL THERAPEUTIC STRATEGY FOR THE TREATMENT OF ALZHEIMER'S DISEASE

Kumar, Amit, Murumkar, Prashant, Kumar, Rajnish, Yadav, Mange Ram, Darreh-Shori, Taher

Journal:

Alzheimer's & Dementia

Year:

2019

File:

PDF, 103 KB

2019